ANASTROZOL 1mg-20 tab
Arimidex (Anastrozole) is an "anti-aromatase" tablet drug that is used by many bodybuilders to prevent gynecomastia and edema, side effects associated with the use of testosterone esters. Anastrozole is the most popular, guaranteed fast way to get rid of aromatization and its effects in the early stages. It works much more effectively than other well-known anti-aromatase drugs such as Tamoxifen or Nolvadex. Aromatase is a key enzyme in estrogen biosynthesis. Anastrozole reduces aromatase activity by about 95% of baseline. Anastrozole has a specific inhibitory effect on aromatase, unlike megestrol acetate or aminoglutethimide. Anastrozole does not affect adrenal steroidogenesis. Anastrozole is able to highly effectively suppress aromatization. The drug is quickly and completely absorbed from the gastrointestinal tract, the maximum concentration of the drug in the blood is reached 2 hours after ingestion on an empty stomach, it is metabolized slowly and, therefore, has a relatively long half-life (40-50 hours), it is excreted mainly in the urine and in smaller quantities. quantities – with bile. The drug should be used 1 time per day for 1 mg (1 tablet). The effect is fully achieved 10-14 days after the start of the drug. It is not recommended to take Anastrozole more than 1 tab per day, as well as for a long time.